Bioactivity:VPC 23019 is a competitive antagonist at the S1P1 and S1P3 receptors (pKi= 7.86 and 5.93, respectively). It is also an agonist at the S1P4 and S1P5 receptors (pEC50= 6.58 and 7.07, respectively).
CAS Nr:
449173-19-7
Purity:
98%
SMILES:
CCCCCCCCC1=CC(=CC=C1)NC(=O)[C@@H](COP(=O)(O)O)N
Formula:
C17H29N2O5P
Molecular weight:
372,4
Pathway:
GPCR/G Protein,GPCR/G Protein
Target:
LPL Receptor,S1P Receptor